Product Information
Molecular Weight 519.2
Purity 99% (TLC: 10% Methanol/methylene chloride; Rf = 0.65)
Recommended Dilutions Potent, selective and widely used inhibitor of PKA (Ki = 48 nM). Cell permeable. Concentration range for cultured cells 30-100 μM: osteoblastic cells, renal proximal tubule cells and Xenopus oocytes.
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2 M.Muroi and T.Suzuki Cell Signal 1993 5 289
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5 A.Azarani et al. J.Biol.Chem. 1995 270 20004
6 A.Azarani et al. J.Biol.Chem. 1995 270 17898
The pharmacological and toxicological properties of this product have not been fully investigated. Exercise caution in use and handling. This product must not be used in humans.